Bisacchi, Gregory S. : rechercher sur Z-Library

Année:

2005

Langue:

english

Fichier:

PDF, 168 KB

english, 2005

Origins of the Quinolone Class of Antibacterials: An Expanded “Discovery Story”

Bisacchi, Gregory S.

Journal:

Keith D. Combrink, H. Belgin Guelgeze, Nicholas A. Meanwell, Bradley C. Pearce, Pi Zulan, Gregory S. Bisacchi, Daniel G. M. Roberts, Paul Stanley, Steven M. Seiler

Année:

2015

Langue:

english

Fichier:

PDF, 433 KB

english, 2015

ChemInform Abstract: 1,2-Benzisothiazol-3-one 1,1-Dioxide Inhibitors of Human Mast Cell Tryptase.

Journal:

ChemInform

Année:

1999

Fichier:

PDF, 29 KB

1999

Synthesis of Potent and Selective 2-Azepanone Inhibitors of Human Tryptase.

Guohua Zhao, Scott A. Bolton, Chet Kwon, Karen S. Hartl, Steven M. Seiler, William A. Slusarchyk, James C. Sutton, Gregory S. Bisacchi

Journal:

ChemInform

Année:

2004

Fichier:

PDF, 83 KB

2004

Synthesis of Potent and Highly Selective Nonguanidine Azetidinone Inhibitors of Human Tryptase.

Gregory S. Bisacchi, et al. et al.

Journal:

ChemInform

Année:

2004

Fichier:

PDF, 84 KB

2004

α-hydroxyamide derived aminodiols as potent inhibitors of hiv protease

Saleem Ahmad, Aaila Ashfaq, Masud Alam, Gregory S. Bisacchi, Ping Chen, Peter T.W. Cheng, Jill A. Greytok, Mark A. Hermsmeier, Pin-Fang Lin, Karen A. Lis, Zoeb Merchant, Toomas Mitt, Mark Skoog, Steve

Journal:

Année:

1995

Langue:

english

Fichier:

PDF, 321 KB

english, 1995

Synthesis of potent and selective 2-azepanone inhibitors of human tryptase

Guohua Zhao, Scott A. Bolton, Chet Kwon, Karen S. Hartl, Steven M. Seiler, William A. Slusarchyk, James C. Sutton, Gregory S. Bisacchi

Journal:

Année:

2004

Langue:

english

Fichier:

PDF, 205 KB

english, 2004

Erratum to “Synthesis of potent and selective 2-azepanone inhibitors of human tryptase” Biorg. Med. Chem. Lett. 14 (2004) 309

Guohua Zhao, ScottA Bolton, Chet Kwon, KarenS Hartl, StevenM Seiler, WilliamA Slusarchyk, JamesC Sutton, GregoryS Bisacchi

Journal:

Année:

2004

Langue:

english

Fichier:

PDF, 72 KB

english, 2004

Synthesis of potent and highly selective nonguanidine azetidinone inhibitors of human tryptase

Gregory S Bisacchi, William A Slusarchyk, Scott A Bolton, Karen S Hartl, Glenn Jacobs, Arvind Mathur, Wei Meng, Martin L Ogletree, Zulan Pi, James C Sutton, Uwe Treuner, Robert Zahler, Guohua Zhao, St

Journal:

Année:

2004

Langue:

english

Fichier:

PDF, 279 KB

english, 2004

(2R, 4S, 5S)-1-(tetrahydro-4-hydroxy-5-methoxy-2-furanyl)thymine: a potent selective inhibitor of herpes simplex thymidine kinase

Choung Un Kim, Peter F. Misco, Bing Y. Luh, Brian Terry, Gregory Bisacchi, Muzammil M. Mansuri

Journal:

Année:

1993

Langue:

english

Fichier:

PDF, 300 KB

english, 1993

Optically active fluorinated cyclobutane nucleoside analogs with potent anti-herpes activity

Saleem Ahmad, Gregory S. Bisacchi, A.Kirk Field, Glenn A. Jacobs, A.Vickie Tuomari, Bridget McGeever-Rubin, Gregory D. Vite, Robert Zahler

Journal:

Année:

1993

Langue:

english

Fichier:

PDF, 301 KB

english, 1993

Solid-phase synthesis and SAR of 4-carboxy-2-azetidinone mechanism-based tryptase inhibitors

James C Sutton, Scott A Bolton, Malcolm E Davis, Karen S Hartl, Bruce Jacobson, Arvind Mathur, Martin L Ogletree, William A Slusarchyk, Robert Zahler, Steven M Seiler, Gregory S Bisacchi

Journal:

Année:

2004

Langue:

english

Fichier:

PDF, 399 KB

english, 2004

Erratum to “Ketene aminal-based lactam derivatives as a novel class of orally active FXa inhibitors” [Bioorg. Med. Chem. Lett. 15 (2005) 5453–5458]

Journal:

Chen, Ping, Cheng, Peter T. W., Alam, Masud, Beyer, Barbara D., Bisacchi, Gregory S., Dejneka, Tamara, Evans, Adelaide J., Greytok, Jill A., Hermsmeier, Mark A., Humphreys, W. Griffith

Année:

2006

Langue:

english

Fichier:

PDF, 55 KB

english, 2006

Aminodiol HIV Protease Inhibitors. Synthesis And Structure−Activity Relationships Of P1/P1‘ Compounds: Correlation between Lipophilicity and Cytotoxicity

Journal:

Année:

1996

Langue:

english

Fichier:

PDF, 982 KB

english, 1996

Amino Diol HIV Protease Inhibitors. 1. Design, Synthesis, and Preliminary SAR

Barrish, Joel C., Gordon, Eric, Alam, Masud, Lin, Pin-Fang, Bisacchi, Gregory S., Chen, Ping, Cheng, Peter T. W., Fritz, Alan W., Greytok, Jill A.

Journal:

Stevens, Robert V., Bisacchi, Gregory S., Goldsmith, Larry, Strouse, C. E.

Année:

1994

Langue:

english

Fichier:

PDF, 1.61 MB

english, 1994

Synthesis of spiro-activated cyclopropanes from alkenes via the irradiation of isopropylidene diazomalonate. A reinvestigation

Journal:

Slusarchyk, William A., Bisacchi, Gregory S., Field, A. Kirk, Hockstein, Deborah R., Jacobs, Glenn A., McGeever-Rubin, Bridget, Tino, Joseph A., Tuomari, A. V., Yamanaka, Gregory A.

Année:

1980

Langue:

english

Fichier:

PDF, 252 KB

english, 1980

Synthesis and antiviral activity of 1-cyclobutyl-5-(2-bromovinyl)uracil nucleoside analogs and related compounds.

Journal:

Bisacchi, Gregory S., Braitman, Abbe, Cianci, Christopher W., Clark, Junius M., Field, A. Kirk, Hagen, Moira E., Hockstein, Deborah R., Malley, Mary F., Mitt, Toomas

Année:

1992

Langue:

english

Fichier:

PDF, 1.10 MB

english, 1992

Synthesis and antiviral activity of enantiomeric forms of cyclobutyl nucleoside analogs

Journal:

Organic Process Research & Development

Année:

1991

Langue:

english

Fichier:

PDF, 981 KB

english, 1991

A Practical Asymmetric Synthesis of the Antiviral Agent Lobucavir, BMS-180194

Singh, Janak, Bisacchi, Gregory S., Ahmad, Saleem, Godfrey,, Jollie D., Kissick, Thomas P., Mitt, Toomas, Kocy, Octavian, Vu, Truc, Papaioannou, Chris G., Wong, Michael K., Heikes, James E., Zahler, R

Journal:

Année:

1998

Langue:

english

Fichier:

PDF, 128 KB

english, 1998

An efficient and remarkably regioselective synthesis of benzocyclobutenones from benzynes and 1,1-dimethoxyethylene

Stevens, Robert V., Bisacchi, Gregory S.

Journal:

Manchester, John I., Buurman, Ed T., Bisacchi, Gregory S., McLaughlin, Robert E.

Année:

1982

Langue:

english

Fichier:

PDF, 2.08 MB

english, 1982

[Annual Reports in Medicinal Chemistry] Annual Reports in Medicinal Chemistry Volume 44 Volume 44 || Chapter 19 Recent Advances in the Inhibition of Bacterial Type II Topoisomerases

Bisacchi, Gregory S.

Année:

2009

Langue:

english

Fichier:

PDF, 1.16 MB

english, 2009

Molecular Determinants of AcrB-Mediated Bacterial Efflux Implications for Drug Discovery

Journal:

Année:

2012

Langue:

english

Fichier:

PDF, 2.14 MB

english, 2012

Discovery of nonbenzamidine factor VIIa inhibitors using a biaryl acid scaffold

Bolton, Scott A., Sutton, James C., Anumula, Rushith, Bisacchi, Gregory S., Jacobson, Bruce, Slusarchyk, William A., Treuner, Uwe D., Wu, Shung C., Zhao, Guohua, Pi, Zulan, Sheriff, Steven, Smirk, Reb

Journal:

Combrink, Keith D., Gülgeze, H. Belgin, Meanwell, Nicholas A., Pearce, Bradley C., Zulan, Pi, Bisacchi, Gregory S., Roberts, Daniel G. M., Stanley, Paul, Seiler, Steven M.

Année:

2013

Langue:

english

Fichier:

PDF, 2.05 MB

english, 2013

1,2-Benzisothiazol-3-one 1,1-Dioxide Inhibitors of Human Mast Cell Tryptase

Journal:

Stevens, Robert V., Bisacchi, Gregory S.

Année:

1998

Langue:

english

Fichier:

PDF, 143 KB

english, 1998

Benzocyclobutenones as synthons for the synthesis of C-11 oxygenated diterpenoids. Application to the total synthesis of (.+-.)-taxodione

Journal:

Bisacchi, Gregory S., Singh, Janak, Godfrey, Jollie D., Kissick, Thomas P., Mitt, Toomas, Malley, Mary F., Di Marco, John D., Gougoutas, Jack Z., Mueller, Richard H., Zahler, Robert

Année:

1982

Langue:

english

Fichier:

PDF, 1.70 MB

english, 1982

Regioselective Coupling of Tetraalkylammonium Salts of 6-Iodo-2-aminopurine to a Cyclobutyl Triflate: Efficient Preparation of Homochiral BMS-180,194, a Potent Antiviral Carbocyclic Nucleoside

Journal: